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KN-62
KN-62是可渗透入细胞的CaM激酶II抑制剂,IC50为0.9 μM,直接与该酶的钙调蛋白结合位点结合,同时还是非竞争性P2X7受体拮抗剂,IC50为15 nM
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KN-62 | MedChemExpress (MCE)
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化合物KN-62 T2694
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KN-62,CaM激酶II抑制剂,127191-97-3,≥98%
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KN-62,127191-97-3,10mM in DMSO
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KN-92
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KN-93 | MedChemExpress (MCE)
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KN-93
KN-93是钙离子/钙调蛋白依赖激酶II(CaMKII)抑制剂,能竞争性阻断钙调蛋白与对应激酶的结合,Ki为370 nM
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KN-93 hydrochloride | MedChemExpress (MCE)
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KN-93 phosphate | MedChemExpress (MCE)
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