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cells from rabbit.?As measured with the [14C]aminopyrine (AP) accumulation method as an index of acid secretion
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(LY2140023) is a high-affinity peptide transporter 1 (PEPT1) substrate with a Km value of ~30 µM. LY2140023 is active
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L-Arg。L-Glutamine 还能抑制缺Arg内皮细胞将L-[14C]Cit转化为L-[14C]Arg。L-Glutamine 可能是通过作用于精氨酸琥珀酸合成酶而不是精氨酸琥珀酸裂解酶来干扰 L-Cit 向 L-Arg 的转化
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%,不影响非HDL胆固醇浓度.与对照组相比,Anacetrapib处理的仓鼠HDL显示ABCG1和SR-B1调节的流出物增多. [14C]Anacetrapib(10 mg/kg,p.o.)给药48 h后,鼠和猴分别恢复~80和90%放射性,但
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NLRP3 抑制剂,抑制 IL-1β 释放的 IC50 为 251.1 nM。NLRP3-IN-10 通过减弱 ASC 斑点形成来抑制 NLRP3炎症小体激活。体外活性: NLRP3-IN-10 (compound 14c) (0.4, 1.6
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|[14c]-ly3214996|6,6-dimethyl-2-(2-((1-methyl-1H-pyrazol-纯度:98%货号:L414043Cas号:1951483-29-6存储温度:-20°C储存产品介绍:Temuterkib
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有效的SGLT1/2抑制剂,用作抗糖尿病剂。体外活性: LX4211 inhibits [14C]AMG uptake with IC50 of 62.0 nM for mouse SGLT1 and 0.6 nM for mouse
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[INN-Latin]|Ro-18-0647|Ro 18-0647/002|Orlistat (Alli, Xenical)|(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl (2S
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Besilate (TAU 284) 是一种选择性可口服的组胺 H1 受体拮抗剂,可用于过敏性鼻炎、过敏性结膜炎、荨麻疹和瘙痒症的研究。激酶实验: Isothermal Titration Calorimetry (ITC
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[14C]acetate without affecting the synthesis of other lipids such as phospholipids (PL), free fatty acids (FFA