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Crenolanib (CP-868596
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DCC-2618
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Imatinib Mesylate (STI571
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PD173074
一种有效的FGFR1抑制剂,IC50约为25 nM,也能抑制VEGFR2,IC50为100-200 nM,作用于FGFR1比作用于PDGFR和c-Src选择性高1000倍左右
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Motesanib
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Tandutinib (MLN518
(MLN518)是一种有效的FLT3拮抗剂,IC50为0.22 μM,同时也抑制PDGFR和c-Kit,对FLT3作用效果比CSF-1R强15到20倍,比FGFR, EGFR和KDR等强100倍以上
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Toceranib
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CP-724714
selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc. Phase 2.
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苏尼替尼
targeting VEGFR2 (Flk-1) and PDGFRβ with IC50 of 80 nM and 2 nM, and also inhibits c-Kit.
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ZM323881
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