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Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, and longer
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KOR antagonist and has the potential as a PET tracer to image KOR in vivo.in vitro: LY2795050 displays full antagonist
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MST1R, FLT3, AXL, MERTK, TEK, ROS1, DDR1/2 and against the serine/threonine kinases MKNK1/2.in vivo: LY2801653
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, the identified small-molecule Haspin inhibitor causes arrest in G2/M and subsequently apoptosis. Importantly, ex vivo
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exposure with AZ20 increases H2AX pan-nuclear staining, indicative of replication stress [2].in vivo: AZ20 induces
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inhibitor both in vitro and in vivo.in vitro: N3PT inhibits transketolase activity in a cell based assay. Competitive
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antagonist at the neurokinin-1 (NK-1) receptor both in vitro and in vivo. In vitro, the binding of NKP608 to bovine retina
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inhibitors. AIC246 exhibits outstanding anti-HCMV activity in vitro and in vivo and currently is undergoing a clinical
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values are 26 and 36000 nM for α4β2 and α7 receptors respectively). Active in vivo
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Reactant used for preparation of fluorescent probes for imaging of tumors in vivo, hypoxia-sensitive